Relistor Drug Information
The drug is an opioid receptor antagonist. It binds to certain receptors and as a result blocks pharmacological actions of opioid drugs. Recently the drug was approved for the treatment of opioid induced constipation (OIC). Relistor is administered mainly to patients with advanced illnesses who take opioids as palliative care to manage pain. Patients can buy Relistor in vials for injection of their contents.
Relistor Drug Dosage
Methylnaltrexone Bromide is administered in subcutaneous injections, in the thigh, upper arm or abdomen. The dosage recommended is once every other day. For patients weighing 38 kg to 62 kg, the dosage recommended is 8 mg. For patients weighing 62 to 114 kg the dosage is 12 mg. For severe renal impairment patients a dose reduction by one half should be made. The appropriate dosage should be determined by the physician. The drug is available as a clear aqueous solution in a dosage of 12 mg. It should be stored at 68 to 77 degrees Fahrenheit and should not be frozen. At North Meds, cheap Relistor comes as a brand drug in the dosage of 12 mg. No generic version can be obtained. Discount Relistor is available in assorted quantities at North Meds.
Side Effects and Precautions for Relistor
Common side effects include flatulence, abdominal pain, dizziness, nausea, diarrhea. More severe side effects comprise confusion or mental clouding. Therefore patients should not do any activity that involves mental sharpness in the 24 hours following injection. Methylnaltrexone Bromide is contraindicated for patients with severe diarrhea lest it may exacerbate their condition, and also for patients with obstructive gastrointestinal tract disorders. Rare cases of gastrointestinal perforations have been reported. In case of diarrhea, discontinue treatment and seek medical consultation. Inform your physician if you have any allergy to opioids. Pregnant and breastfeeding women should avoid using the drug.
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